{"id":23116,"date":"2025-04-13T17:39:10","date_gmt":"2025-04-13T17:39:10","guid":{"rendered":"https:\/\/globalsourcechemicals.com\/?post_type=product&#038;p=23116"},"modified":"2025-10-03T19:21:36","modified_gmt":"2025-10-03T19:21:36","slug":"etizolam-1-mg-pelete","status":"publish","type":"product","link":"https:\/\/globalsourcechemicals.com\/sl\/trgovina\/prepovedano\/etizolam-1-mg-pelete\/","title":{"rendered":"Etizolam 1 mg peleti"},"content":{"rendered":"<h1><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam 1 mg peleti \u2013 tienodiazepinska raziskovalna formulacija laboratorijske kakovosti<\/span><\/span><\/strong><\/h1>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pregled zdravila Etizolam<\/span><\/span><\/h2>\n<p><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam je tienodiazepinski analog z mo\u010dnimi anksioliti\u010dnimi, sedativnimi in mi\u0161i\u010dno-relaksantnimi lastnostmi. Te 1 mg pelete so bile razvite za kontrolirane \u0161tudije interakcij receptorjev GABA-A in nevrofarmakolo\u0161kih procesov. <\/span><\/span><a href=\"https:\/\/globalsourcechemicals.com\/sl\/trgovina\/lisergamidi\/1vlsd\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">1V-LSD 150 MCG pivniki<\/span><\/span><\/a><\/p>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Zna\u010dilnosti izdelka<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Natanko 1 mg etizolama na peleto (variacija \u00b12%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Formulirano z mikrokristalno celulozo<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Fotostabilna in vlagoodporna embala\u017ea<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Serija preverjena za:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u010cistost HPLC (\u226598%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Preverjanje identitete MS<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Izena\u010denost te\u017ee in velikosti<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Farmakolo\u0161ki profil<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Visoka afiniteta za receptorje GABA-A<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Selektivna vezava na podtipe \u03b11\u2013\u03b15<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Farmakolo\u0161ko delovanje:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Anksiolitik<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pomirjevalo<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Mi\u0161i\u010dni relaksant<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Kraj\u0161i razpolovni \u010das izlo\u010danja kot pri klasi\u010dnih benzodiazepinih<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Podro\u010dja uporabe v raziskavah<\/span><\/span><\/h2>\n<ol>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Nevrofarmakologija<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Interakcije receptorjev GABA-A<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Alosteri\u010dna modulacija<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Specifi\u010dnost podtipa<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Primerjalna analiza<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Primerjava strukture in aktivnosti z benzodiazepini<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Raziskave presnovnih poti<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Vedenjska znanost<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Modeli anksioznosti (npr. EPM, OFT)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Cikli spanja in budnosti<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Zatiranje konvulzij<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ol>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Tehni\u010dne specifikacije<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Premer pelete: 2,5 mm \u00b1 0,1 mm<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Te\u017ea: 10 mg \u00b1 0,5 mg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Barva: \u010cisto bela<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Topnost: &gt;5 mg\/ml v etanolu (96%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Tali\u0161\u010de: 146\u2013148 \u00b0C<\/span><\/span><\/li>\n<\/ul>\n<h3><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Profil stabilnosti<\/span><\/span><\/h3>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Rok uporabnosti: 36 mesecev pri 15\u201325 \u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Svetlobna obstojnost: &lt;1% degradacija\/leto<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Vsebnost vlage: &lt;0,51 TP3T (Karl Fischer)<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Navodila za odmerjanje (samo za referenco)<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">In vitro: 10\u20131000 nM<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Predklini\u010dno: 0,05\u20130,5 mg\/kg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Vedenjski modeli: 0,1\u20131,0 mg\/kg<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Informacije o varnosti in shranjevanju<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Hranite v embala\u017ei, ki ne prepu\u0161\u010da svetlobe<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Relativna vla\u017enost &lt;40%<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Temperatura med 15\u201325 \u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Zdru\u017eljivo s PBS, NaCl 0.9% <\/span><\/span><a href=\"https:\/\/globalsourcechemicals.com\/sl\/trgovina\/pellets\/o-dsmt-50-mg-pelete\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">O-DSMT 50 mg peleti<\/span><\/span><\/a><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Dokumentacija ob dostavi<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Potrdilo o originalnosti z:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u010cistost<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u010cas zadr\u017eevanja<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Masovna identifikacija<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Varnostni list (SDS) v skladu z GHS<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Tehni\u010dni list z:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Podatki o stabilnosti<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Predlogi eksperimentalne zasnove<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Analiza topnosti<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p><em><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Samo za znanstvene namene. Ni primerno za medicinsko, diagnosti\u010dno ali \u010dlove\u0161ko uporabo. <\/span><\/span><a href=\"https:\/\/globalsourcechemicals.com\/sl\/trgovina\/top-10-research-chemicals\/oksidacija-kaluje\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Oksidiranje Caluanie Muelear<\/span><\/span><\/a><\/em><\/p>","protected":false},"excerpt":{"rendered":"<h2><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam pellets properties<\/span><\/span><\/span><\/span><\/h2>\n<p><strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Synonym<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 4-(2-chlorophenyl)-2-ethyl-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">CAS Number<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 40054-69-1 <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Formula<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : C17H15ClN4S <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Molar mass<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 342.8 g\/mol <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Purity<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : \u2265 99%<\/span><\/span><\/span><\/span><\/p>\n","protected":false},"featured_media":28491,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[82],"product_cat":[488],"product_tag":[917,326],"class_list":{"0":"post-23116","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_brand-research-chemical","7":"product_cat-verboden","8":"product_tag-etizolam","9":"product_tag-nl","11":"first","12":"instock","13":"taxable","14":"shipping-taxable","15":"purchasable","16":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/product\/23116","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/comments?post=23116"}],"version-history":[{"count":6,"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/product\/23116\/revisions"}],"predecessor-version":[{"id":28492,"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/product\/23116\/revisions\/28492"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/media\/28491"}],"wp:attachment":[{"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/media?parent=23116"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/product_brand?post=23116"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/product_cat?post=23116"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sl\/wp-json\/wp\/v2\/product_tag?post=23116"}],"curies":[{"name":"delovni 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