{"id":23662,"date":"2025-04-13T17:40:11","date_gmt":"2025-04-13T17:40:11","guid":{"rendered":"https:\/\/globalsourcechemicals.com\/?post_type=product&#038;p=23662"},"modified":"2025-10-03T07:21:02","modified_gmt":"2025-10-03T07:21:02","slug":"flualprazolam-1-mg-pelety","status":"publish","type":"product","link":"https:\/\/globalsourcechemicals.com\/sk\/obchod\/zakazane\/flualprazolam-1-mg-pelety\/","title":{"rendered":"Flualprazolam 1 MG pelety"},"content":{"rendered":"<div id=\"content_tab_description\" class=\"tab-content tab-description\">\n<div class=\"tab-content-inner\">\n<div class=\"tab-content-scroll\">\n<h1><strong>Flualprazolam 1 MG pelety \u2013 v\u00fdskumn\u00e1 zl\u00fa\u010denina so silnou benzodiazep\u00ednovou aktivitou<\/strong><\/h1>\n<p><strong>N\u00e1zov produktu:<\/strong> Flualprazolam 1 MG pelety<br \/>\n<strong>Chemick\u00e1 trieda:<\/strong> Triazolobenzodiazep\u00edn<br \/>\n<strong>Vzorec:<\/strong> C17H12ClFN4<br \/>\n<strong>Molekulov\u00e1 hmotnos\u0165:<\/strong> 342,8 g\/mol<br \/>\n<strong>\u010distota:<\/strong> \u2265 98% (overen\u00e9 HPLC)<br \/>\n<strong>Formul\u00e1r:<\/strong> Mikrolisovan\u00e9 pelety s hmotnos\u0165ou 1 mg<\/p>\n<hr \/>\n<h2><strong>Popis<\/strong><\/h2>\n<p>Flualprazolam je siln\u00e1 zl\u00fa\u010denina benzodiazep\u00ednov a je \u0161truktur\u00e1lne pr\u00edbuzn\u00e1 alprazolamu (Xanax), pri\u010dom charakteristick\u00fdm znakom je pridanie at\u00f3mu flu\u00f3ru k fenylov\u00e9mu kruhu. T\u00e1to jemn\u00e1 chemick\u00e1 modifik\u00e1cia zvy\u0161uje afinitu k receptorom GABAA, \u010do vedie k zv\u00fd\u0161enej \u00fa\u010dinnosti a dlh\u0161iemu trvaniu \u00fa\u010dinku.<\/p>\n<p>Pelety Flualprazolam 1 MG s\u00fa presne d\u00e1vkovan\u00e9 a ur\u010den\u00e9 v\u00fdhradne na <strong>analytick\u00e9 \u00fa\u010dely, referen\u010dn\u00fd v\u00fdskum a laborat\u00f3rna anal\u00fdza<\/strong>Nie je ur\u010den\u00e9 na \u013eudsk\u00fa spotrebu.<\/p>\n<hr \/>\n<h2><strong>Aplik\u00e1cie a v\u00fdskumn\u00e9 \u00fa\u010dely<\/strong><\/h2>\n<ul>\n<li>Farmakodynamick\u00e9 \u0161t\u00fadie GABAergn\u00fdch interakci\u00ed<\/li>\n<li>\u0160t\u00fadie v\u00e4zby na receptory a porovnanie s in\u00fdmi triazolobenzodiazep\u00ednmi<\/li>\n<li>Behavior\u00e1lne \u0161t\u00fadie na zvierac\u00edch modeloch za kontrolovan\u00fdch podmienok<\/li>\n<li>Anal\u00fdzy stability a rozpustnosti v r\u00f4znych rozp\u00fa\u0161\u0165adl\u00e1ch<\/li>\n<li>Referencia v toxikologick\u00fdch alebo analytick\u00fdch laborat\u00f3ri\u00e1ch (kalibr\u00e1cia GC-MS\/LC-MS)<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>V\u00fdhody pre v\u00fdskumn\u00edkov<\/strong><\/h2>\n<p>\u2705 <strong>Vysok\u00e1 \u00fa\u010dinnos\u0165<\/strong> \u2013 Pre badate\u013en\u00e9 \u00fa\u010dinky v experiment\u00e1lnych podmienkach je potrebn\u00e1 n\u00edzka d\u00e1vka<br \/>\n\u2705 <strong>Stabiln\u00fd tvar peliet<\/strong> \u2013 Jednoduch\u00e9 d\u00e1vkovanie a skladovanie<br \/>\n\u2705 <strong>Laborat\u00f3rne testovan\u00e1 \u010distota<\/strong> \u2013 Zaru\u010den\u00e1 konzistentnos\u0165 pre reprodukovate\u013en\u00e9 v\u00fdsledky v\u00fdskumu<\/p>\n<hr \/>\n<h2><strong>Nev\u00fdhody a rizik\u00e1<\/strong><\/h2>\n<p>\u26a0\ufe0f <strong>Ve\u013emi siln\u00fd<\/strong> \u2013 Aj minim\u00e1lne odch\u00fdlky v d\u00e1vkovan\u00ed m\u00f4\u017eu v\u00fdrazne ovplyvni\u0165 v\u00fdsledok experimentov<br \/>\n\u26a0\ufe0f <strong>Dlhotrvaj\u00faci \u00fa\u010dinok<\/strong> \u2013 Po opakovanom pod\u00e1van\u00ed m\u00f4\u017ee vies\u0165 k akumul\u00e1cii v zvierac\u00edch modeloch<br \/>\n\u26a0\ufe0f <strong>Potreba podmienen\u00e9ho skladovania<\/strong> \u2013 Skladujte najlep\u0161ie pri teplote do 25 \u00b0C, v suchu a tme<\/p>\n<hr \/>\n<h2><strong>Pou\u017eitie a laborat\u00f3rne pokyny<\/strong><\/h2>\n<ul>\n<li><strong>Odpor\u00fa\u010dan\u00e9 laborat\u00f3rne d\u00e1vkovanie:<\/strong> Pri in vitro testoch za\u010dnite s d\u00e1vkou 0,25 \u2013 0,5 mg. Bez kalibr\u00e1cie neprekra\u010dujte t\u00fato d\u00e1vku.<\/li>\n<li><strong>Rozpustnos\u0165:<\/strong> \u013dahko rozpustn\u00fd v etanole, DMSO a propyl\u00e9nglykole<\/li>\n<li><strong>Podmienky skladovania:<\/strong> Skladujte vo vzduchotesnej n\u00e1dobe, v chlade a mimo dosahu priameho slne\u010dn\u00e9ho \u017eiarenia<\/li>\n<li><strong>Manipul\u00e1cia:<\/strong> Pri manipul\u00e1cii s pr\u00e1\u0161kom alebo roztokom noste rukavice, ochrann\u00e9 okuliare a pracujte pod digestorom.<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>\u010casto kladen\u00e9 ot\u00e1zky (FAQ)<\/strong><\/h2>\n<h3>\u2753 <em>Je Flualprazolam leg\u00e1lny v Holandsku alebo Belgicku?<\/em><\/h3>\n<p>\u27a1\ufe0f Pr\u00e1vny status sa l\u00ed\u0161i. V\u017edy si overte najnov\u0161ie miestne predpisy. Konzum\u00e1cia je vo v\u0161eobecnosti zak\u00e1zan\u00e1, ale m\u00f4\u017ee by\u0165 povolen\u00e1 na analytick\u00e9 testovanie.<\/p>\n<h3>\u2753 <em>M\u00f4\u017eem pou\u017ei\u0165 Flualprazolam na v\u00fdskum sp\u00e1nku alebo \u00fazkosti?<\/em><\/h3>\n<p>\u27a1\ufe0f Len v pr\u00edsne kontrolovanom laborat\u00f3rnom prostred\u00ed a v\u00fdlu\u010dne na ne\u013eudsk\u00fdch modeloch alebo v \u0161t\u00fadi\u00e1ch chemick\u00fdch interakci\u00ed.<\/p>\n<h3>\u2753 <em>Ako dlho zost\u00e1va Flualprazolam stabiln\u00fd pri izbovej teplote?<\/em><\/h3>\n<p>\u27a1\ufe0f V such\u00fdch a tmav\u00fdch podmienkach zost\u00e1va stabiln\u00fd minim\u00e1lne 12 mesiacov pri teplote 20\u201325 \u00b0C.<\/p>\n<h3>\u2753 <em>Existuje skr\u00ed\u017een\u00e1 rezistencia s in\u00fdmi benzodiazep\u00ednmi?<\/em><\/h3>\n<p>\u27a1\ufe0f \u00c1no, flualprazolam vykazuje prekr\u00fdvaj\u00face sa v\u00e4zbov\u00e9 profily s in\u00fdmi l\u00e1tkami, ako s\u00fa alprazolam a klonazolam.<\/p>\n<hr \/>\n<h2><strong>S\u00fahrn laborat\u00f3rnej spr\u00e1vy<\/strong><\/h2>\n<table>\n<thead>\n<tr>\n<th>Parameter<\/th>\n<th>Hodnota<\/th>\n<\/tr>\n<\/thead>\n<tbody>\n<tr>\n<td><strong>\u010c\u00edslo \u0161ar\u017ee<\/strong><\/td>\n<td>FLPZ-0725<\/td>\n<\/tr>\n<tr>\n<td><strong>\u010cistota (HPLC)<\/strong><\/td>\n<td>99,3%<\/td>\n<\/tr>\n<tr>\n<td><strong>Vzh\u013ead<\/strong><\/td>\n<td>Biely kry\u0161talick\u00fd pr\u00e1\u0161ok (zlisovan\u00fd do peliet)<\/td>\n<\/tr>\n<tr>\n<td><strong>Bod topenia<\/strong><\/td>\n<td>225 \u2013 230 \u00b0C<\/td>\n<\/tr>\n<tr>\n<td><strong>Identifik\u00e1cia<\/strong><\/td>\n<td>Potvrden\u00e9 NMR a MS<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<hr \/>\n<h2><strong>POZOR<\/strong><\/h2>\n<p><strong>Nie je ur\u010den\u00e9 na \u013eudsk\u00fa spotrebu ani na lek\u00e1rske pou\u017eitie. Len na profesion\u00e1lny v\u00fdskum v kvalifikovan\u00fdch laborat\u00f3ri\u00e1ch.<\/strong><\/p>\n<\/div>\n<\/div>\n<\/div>","protected":false},"excerpt":{"rendered":"<h3><span data-sheets-value=\"{\" data-sheets-userformat=\"{\"><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Flualprazolam Pellets Properties<\/span><\/span><\/span><\/h3>\n<p><strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Synonym:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> Fluclazolam <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">CAS Number:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 28910-91-0 <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Formula:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 8-chloro-6-(2-fluorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Molar mass:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 326.8 g\/mol <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Purity:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> &gt;97%<\/span><\/span><\/p>\n","protected":false},"featured_media":27882,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[488],"product_tag":[326],"class_list":{"0":"post-23662","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-verboden","7":"product_tag-nl","9":"first","10":"instock","11":"taxable","12":"shipping-taxable","13":"purchasable","14":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/product\/23662","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/comments?post=23662"}],"version-history":[{"count":4,"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/product\/23662\/revisions"}],"predecessor-version":[{"id":25752,"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/product\/23662\/revisions\/25752"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/media\/27882"}],"wp:attachment":[{"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/media?parent=23662"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/product_brand?post=23662"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/product_cat?post=23662"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/sk\/wp-json\/wp\/v2\/product_tag?post=23662"}],"curies":[{"name":"pracovn\u00fd list","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}