2C-B-FLY 10 mg peleta
2C-B-FLY 10 mg peleta Raspon cijena: od €49.95 do €199.95
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Flunitrazolam 0,25 mg pelete

Raspon cijena: od €6.00 do €180.43

Flunitrazolam 0.25 mg Pellets – Precision Dosed Benzodiazepine Analogue for Scientific Research

Introduction to Flunitrazolam

Flunitrazolam is a highly potent triazolo-benzodiazepine-like compound with distinct pharmacological properties. These 0.25 mg pellets were specifically developed for controlled scientific research into GABAergic neurotransmission and related neurological processes.

Critical Quality Characteristics

  • Točno doziranje : Each pellet contains exactly 0.25 mg Flunitrazolam (±2% variation)
  • Advanced pharmaceutical formulation : Microcrystalline cellulose matrix for optimal bioavailability
  • Stabilan sastav : Protected against photodegradation and moisture absorption
  • Rigorous quality control : Each production batch is subject to:
    • HPLC analysis (purity ≥98%)
    • Mass spectrometry confirmation
    • Uniformity control of weight and diameter

Pharmacodynamic Properties

Flunitrazolam exhibits characteristic properties:

  • Extremely high potency : Active in nanomolar concentrations
  • Selective GABA-A receptor modulation :
    • Strong binding to α1, α2, and α3 subunit-containing receptors
    • Amplification of chloride ion current
  • Pronounced pharmacological effects :

Scientific Research Applications

Particularly valuable for:

  1. Neurofarmakološke studije :
    • GABAergic signal transduction mechanisms
    • Receptor subtype specificity
    • Allosteric modulation processes
  2. Komparativna farmakologija :
    • Potency comparison with classical benzodiazepines
    • Structural-activity relationships within triazolobenzodiazepines
  3. Behavioral Neuroscience :
    • Anxiety-related behavioral paradigms
    • Sleep-wake cycle research
    • Seizure inhibition studies

Tehničke specifikacije

  • Fizičke karakteristike :
    • Diameter: 2.0mm ± 0.1mm
    • Weight: 8 mg ± 0.5 mg per pellet
    • Boja: Čisto bijela
    • Topljivost: >5 mg/ml u etanolu (96%)
  • Stability parameters :
    • Shelf life: 36 months at 15-25°C (in original packaging)
    • Light sensitivity: Photodegradation <1% per year (stored in the dark)
    • Moisture content: <0.5% (Karl Fischer method)

Research dosage

Samo za znanstvenu referencu:

  • Studije in vitro : 1-100 nM concentrations
  • Preclinical evaluations : 0.01-0.1 mg/kg body weight
  • Bihevioralne studije : 0.02-0.2 mg/kg (model-dependent). 1V-LSD 150 MCG upijajućih papira

Safety and Storage Protocols

  • Stability guarantee : Under controlled conditions
  • Compatibility studies : Verified with:
    • Physiological saline solution (0.9% NaCl)
    • Phosphate buffer (PBS, pH 7.4)
    • Dimethyl sulfoxide (DMSO)
  • Storage requirements :
    • Primary packaging: Light-blocking glass
    • Secondary packaging: Oxygen absorbing material
    • Temperature range: 15-25°C

Quality documentation

With every order you will receive:

  1. Analytical Certificate of Analysis including:
  • HPLC chromatogram
  • Mass spectrum
  • Purity percentage
  • Heavy metal analysis
  1. Extended Safety Data Sheet according to GHS standard
  2. Technical Support Documentation :
  • Solubility data
  • Profil stabilnosti
  • Proposed research protocols

These pellets are intended solely for scientific research by qualified professionals in controlled laboratory environments. Not intended for diagnostic or therapeutic use. 1cP-LSD 150 MCG Art Blotters

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