Etizolam 1 MG Micro Pellets – Precision Dosing for Research Purposes
Nom du produit: Etizolam 1 mg Micro Pellets
Active Substance: Étizolam
Classe chimique : Thienodiazepine (benzodiazepine analogue)
Formule moléculaire: C17H15ClN4S
Masse moléculaire: 342.85 g/mol
Formulaire: Micro Pellets (submillimeter size)
Dosage: 1 mg per pellet
Conditionnement: 10 / 25 / 50 / 100 pellets
Application: For laboratory and analytical research only
🔬 What is Etizolam?
Etizolam is a thienodiazepine compound structurally related to traditional benzodiazepines. It is known for its potent GABA-A receptor agonism , which produces anxiolytic, sedative, and muscle relaxant effects . In analytical studies, Etizolam is being evaluated for its receptor binding profile , stability , et structural-activity relationships (SAR) within the benzodiazepine family.
Le micro pellet shape offers exceptional precision dosing and reproducibility , ideal for fine-mesh laboratory applications and storage.
✅ Applications en recherche
- Neuroreceptor analysis: GABA-A modulation in vitro
- Etude de l'activité structurale (SAR) : Comparison with classical benzos (diazepam, alprazolam)
- Stability studies: Under the influence of temperature, moisture and light
- Pharmacokinetics (preclinical): In vivo simulations under ethical protocol
- Analytical reference substance: LC-MS, HPLC, NMR
⚠️ Prudence: Not suitable for human or animal consumption. For professional research purposes only.
⚠️ Risques et limites
- Very potent in low doses – incorrect use can be dangerous
- Dependency potential with abuse
- Possible regulation in EU/US – considered a controlled substance in some countries
- Not intended for recreational use or self-experimentation
- May cause drowsiness or motor disorders if handled incorrectly
🧪 Détails du laboratoire
| Caractéristiques | Spécification |
|---|---|
| substance active | Etizolam (≥99% purity – HPLC, GC-MS) |
| Formulaire | Micro pellets (approximately 0.6–0.8 mm diameter) |
| Dosage | 1 mg per pellet |
| Couleur | Blanc à gris clair |
| Stabilité | ≥ 24 months when stored correctly |
| Solubilité | Soluble in ethanol, DMSO, acetonitrile |
| Conseils de stockage | Dark, dry, cool (2–8 °C) |
| COA | Disponible sur demande |
💡 Cas d'utilisation recommandés
| Research area | Application |
|---|---|
| Études de liaison aux récepteurs | GABA-A response in different subtypes |
| Chimie analytique | Reference in HPLC or LC-MS equipment |
| Stability testing | Under stressful conditions in the laboratory |
| Recherche SAR | Comparison with other thienodiazepines |
❓ Foire aux questions (FAQ)
1. What is the difference between a micro pellet and a regular pellet?
Micro pellets are much smaller (submillimeter size) and designed for highly accurate dosing and rapid dissolution during analytical processes.
2. Is Etizolam legal?
That varies by country. In some regions, Etizolam is a controlled substance . Always check the regulations in your country before ordering or using it.
3. Is this product suitable for human consumption?
Non. Ces granulés sont intended for laboratory use only . Use on humans or animals is prohibited and potentially dangerous.
4. How should I store the pellets?
Store them in a tightly closed, dry container at 2–8°C , à l'abri de la lumière et de l'humidité.
5. Is a Certificate of Analysis available?
Oui, un COA (Certificat d'analyse) is available upon request for each batch. This includes HPLC data, purity, and lot number.
📦 Présentation du produit
| Fonctionnalité | Spécification |
|---|---|
| Nom du produit | Microgranules d'étizolam 1 mg |
| Formulaire | Submillimeter pressed pellets |
| Dosage | 1 mg per pellet |
| Conditionnement | 10 / 25 / 50 / 100 pellets |
| Pureté | ≥99% |
| Usage | Pour usage en laboratoire uniquement |
| Conditions de stockage | Frais, sec et à l'abri de la lumière |
| Statut juridique | Selon la région |
| COA | Disponible par lot |
| 5 étoiles | 67 | 67% |
| 4 étoiles | 33 | 33% |
| 3 étoiles | 0% | |
| 2 étoiles | 0% | |
| 1 étoile | 0% |
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