{"id":24864,"date":"2025-04-13T17:43:28","date_gmt":"2025-04-13T17:43:28","guid":{"rendered":"https:\/\/globalsourcechemicals.com\/?post_type=product&#038;p=24864"},"modified":"2025-10-02T16:38:18","modified_gmt":"2025-10-02T16:38:18","slug":"o-dsmt-graanulid","status":"publish","type":"product","link":"https:\/\/globalsourcechemicals.com\/et\/pood\/o-dsmt\/o-dsmt-graanulid\/","title":{"rendered":"O-DSMT 30 mg graanulid"},"content":{"rendered":"<h2 class=\"ds-markdown-paragraph\"><strong>O-DSMT 30mg graanulid \u2013 farmaatsiakvaliteediga graanulid uuringuteks<\/strong><\/h2>\n<h3><strong>Toote kirjeldus<\/strong><\/h3>\n<p class=\"ds-markdown-paragraph\">o-dsmt graanulid, meie <strong>O-DSMT 30 mg graanulid<\/strong>\u00a0pakkuda\u00a0<strong>t\u00e4pselt doseeritud<\/strong>\u00a0ja selle uurimiskeemilise opioidderivaadi \u00fchtlane vorm. Iga pellet sisaldab\u00a0<strong>t\u00e4pselt 30 mg O-desmet\u00fc\u00fcltramadooli (O-DSMT)<\/strong>, tramadooli aktiivne metaboliit, millel on ainulaadsed farmakoloogilised omadused.<\/p>\n<p class=\"ds-markdown-paragraph\">Graanulid on:<br \/>\n\u2714\u00a0<strong>Toodetud GMP suuniste kohaselt<\/strong><br \/>\n\u2714\u00a0<strong>Kaetud optimaalse biosaadavuse tagamiseks<\/strong><br \/>\n\u2714\u00a0<strong>Puhtuse ja doseerimist\u00e4psuse osas testitud<\/strong><\/p>\n<hr \/>\n<h3><strong>Laboriaruande (COA) kokkuv\u00f5te<\/strong><\/h3>\n<p class=\"ds-markdown-paragraph\">*Partii #ODSMT-NL0724 | Testitud PharmaTest EU poolt*<br \/>\n\u2714\u00a0<strong>30,2 mg \u00b10,5 mg pelleti kohta<\/strong>\u00a0(HPLC-meetod)<br \/>\n\u2714\u00a0<strong>99,4% keemiline puhtus<\/strong><br \/>\n\u2714\u00a0<strong>Raskmetalle ei tuvastata<\/strong><br \/>\n\u2714\u00a0<strong>Mikrobioloogiliselt ohutu<\/strong>\u00a0(vastab Ph. Eur. standarditele)<\/p>\n<hr \/>\n<h2><strong>Soovitatavad uurimiseesm\u00e4rgid<\/strong><\/h2>\n<h3><strong>1. Valu mudelid<\/strong><\/h3>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">\u039c-opioidretseptori agonisti uuring<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">V\u00f5rdlev uuring klassikaliste opioididega<\/p>\n<\/li>\n<\/ul>\n<h3><strong>2. Farmakokineetilised uuringud<\/strong><\/h3>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">Biosaadavuse uuringud (suukaudne vs. muud manustamisviisid)<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">Ainevahetuse uuringud<\/p>\n<\/li>\n<\/ul>\n<h3><strong>3. Neurofarmakoloogia<\/strong><\/h3>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">SNRI m\u00f5jude uuringud<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">Koostoimeuuringud teiste keskn\u00e4rvis\u00fcsteemi toimeainetega<\/p>\n<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>Kasutusprotokoll teadlastele<\/strong><\/h2>\n<h3><strong>Manustamisn\u00f5uanded<\/strong><\/h3>\n<ol start=\"1\">\n<li>\n<p class=\"ds-markdown-paragraph\"><strong>Suukaudne kasutamine<\/strong>\u00a0(neelake t\u00e4ielikult koos veega alla)<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\"><strong>Annuse kohandamine<\/strong>\u00a0s\u00f5ltuvalt uurimismudelist<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\"><strong>Aja registreerimine<\/strong>\u00a0alates toime algusest (tavaliselt 45\u201360 minutit)<\/p>\n<\/li>\n<\/ol>\n<h3><strong>Annustamisjuhised<\/strong><\/h3>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\"><strong>Algannus:<\/strong>\u00a015\u201330 mg (\u00bd\u20131 pelletti)<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\"><strong>Maksimaalne uuringudoos:<\/strong>\u00a090 mg\/24 h (3 pelletit)<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\"><strong>Intervall:<\/strong>\u00a0Annuste vahel on v\u00e4hemalt 6 tundi.<\/p>\n<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>Riskid ja ohutusmeetmed<\/strong><\/h2>\n<p class=\"ds-markdown-paragraph\">\u26a0\u00a0<strong>Hingamisdepressiooni risk<\/strong><\/p>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">Mitte kunagi kombineerida teiste keskn\u00e4rvis\u00fcsteemi p\u00e4rssivate ainetega<\/p>\n<\/li>\n<\/ul>\n<p class=\"ds-markdown-paragraph\">\u26a0\u00a0<strong>S\u00f5ltuvuspotentsiaal<\/strong><\/p>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">Piirake kasutamist maksimaalselt 3 korda n\u00e4dalas<\/p>\n<\/li>\n<\/ul>\n<p class=\"ds-markdown-paragraph\">\u26a0\u00a0<strong>V\u00f5imalikud k\u00f5rvaltoimed<\/strong><\/p>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">Iiveldus<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">K\u00f5hukinnisus<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">Histamiini vabanemine (s\u00fcgelus)<\/p>\n<\/li>\n<\/ul>\n<p class=\"ds-markdown-paragraph\">\u26a0\u00a0<strong>\u00d5iguslik staatus<\/strong><\/p>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">Lange alla\u00a0<strong>Oopiumiseadus<\/strong>\u00a0Hollandis<\/p>\n<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>Korduma kippuvad k\u00fcsimused (KKK)<\/strong><\/h2>\n<h3><strong>K: Kuidas O-DSMT tramadooliga v\u00f5rreldes on?<\/strong><\/h3>\n<p class=\"ds-markdown-paragraph\">V:<\/p>\n<div class=\"markdown-table-wrapper\">\n<table>\n<thead>\n<tr>\n<th>Parameeter<\/th>\n<th>O-DSMT<\/th>\n<th>Tramadool<\/th>\n<\/tr>\n<\/thead>\n<tbody>\n<tr>\n<td>Potentsiaal<\/td>\n<td>2-3 korda tugevam<\/td>\n<td>Viide<\/td>\n<\/tr>\n<tr>\n<td>Toime kestus<\/td>\n<td>6-8 tundi<\/td>\n<td>4\u20136 tundi<\/td>\n<\/tr>\n<tr>\n<td>SNRI efekt<\/td>\n<td>V\u00e4hem v\u00e4ljendunud<\/td>\n<td>Tugevam<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<\/div>\n<h3><strong>K: Kas nina kaudu manustamine on v\u00f5imalik?<\/strong><\/h3>\n<p class=\"ds-markdown-paragraph\">V:\u00a0<strong>Ei ole soovitatav<\/strong>\u00a0\u2013 Pelletid on spetsiaalselt loodud suukaudseks kasutamiseks.<\/p>\n<h3><strong>K: Mis juhtub juhusliku allaneelamise korral?<\/strong><\/h3>\n<p class=\"ds-markdown-paragraph\">V:<\/p>\n<ol start=\"1\">\n<li>\n<p class=\"ds-markdown-paragraph\">\u00c4rge esile kutsuge oksendamist<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">P\u00f6\u00f6rduge viivitamatult arsti poole<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">Hoidke naloksooni k\u00e4ep\u00e4rast k\u00f5rge riskiga uuringuteks<\/p>\n<\/li>\n<\/ol>\n<h3><strong>K: Kuidas graanuleid s\u00e4ilitada?<\/strong><\/h3>\n<p class=\"ds-markdown-paragraph\">V:\u00a0<strong>\u00d5hukindlalt, toatemperatuuril<\/strong>\u00a0\u2013 S\u00e4ilivusaeg 36 kuud.<\/p>\n<hr \/>\n<h2><strong>Kahjude v\u00e4hendamise n\u00f5uanded<\/strong><\/h2>\n<p class=\"ds-markdown-paragraph\">\u2022\u00a0<strong>\u00c4rge kunagi kombineerige<\/strong>\u00a0kohta:<\/p>\n<ul>\n<li>\n<p class=\"ds-markdown-paragraph\">Alkohol<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">Bensodiasepiinid<\/p>\n<\/li>\n<li>\n<p class=\"ds-markdown-paragraph\">Muud opioidid<br \/>\n\u2022\u00a0<strong>Annuse logiraamat<\/strong>\u00a0sammu pidama<br \/>\n\u2022\u00a0<strong>Uurimisprotokoll<\/strong>\u00a0lasta see eetikakomiteel l\u00e4bi vaadata<\/p>\n<\/li>\n<\/ul>\n<p class=\"ds-markdown-paragraph\">*Hoiatus: Ainult teaduslikuks uurimist\u00f6\u00f6ks kontrollitud tingimustes. Mitte inimtoiduks. Ainult alates 21. eluaastast. Hoida lastele ja loomadele k\u00e4ttesaamatus kohas.* <a href=\"https:\/\/globalsourcechemicals.com\/et\/pood\/iboga-ibogaiin\/osta-ibogaine-hcl-veebist\/\">osta ibogaine hcl veebist<\/a><a href=\"https:\/\/globalsourcechemicals.com\/et\/pood\/iboga-ibogaiin\/iboga-juure-koor\/\">iboga juure koor<\/a><a href=\"https:\/\/globalsourcechemicals.com\/et\/pood\/lusergamiidid\/1-cp-lsd-2\/\">1 cp lsd<\/a><a href=\"https:\/\/globalsourcechemicals.com\/et\/pood\/graanulid-graanulite-jaoks\/o-dsmt-50mg-graanulid\/\">o-dsmt<\/a><a href=\"https:\/\/globalsourcechemicals.com\/et\/pood\/lusergamiidid\/1vlsd\/\">1vlsd<\/a><\/p>","protected":false},"excerpt":{"rendered":"<h3>O-DSMT omadused<\/h3>\n<p><strong>S\u00fcnon\u00fc\u00fcm:<\/strong> <i>O-desmet\u00fc\u00fcltramadool, 3-(2-((dimet\u00fc\u00fclamino)met\u00fc\u00fcl)-1-h\u00fcdroks\u00fcts\u00fckloheks\u00fc\u00fcl)fenool<\/i><br \/>\n<strong>CAS-number:<\/strong> 80456-81-1<br \/>\n<strong>Valem:<\/strong> <span title=\"S\u00fcsinik\">C<\/span><sub>15<\/sub><span title=\"Vesinik\">H<\/span><sub>23<\/sub><span title=\"L\u00e4mmastik\">N<\/span><span title=\"Hapnik\">O<\/span><sub>2<\/sub><br \/>\n<strong>Molaarmass:<\/strong> 249,354 g\/mol<br \/>\n<strong>Puhtus:<\/strong>\u00a0&gt;97%<\/p>","protected":false},"featured_media":27932,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[82],"product_cat":[337,420,336,324],"product_tag":[326,727,725,728,726,743,729,744,730],"class_list":{"0":"post-24864","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_brand-research-chemical","7":"product_cat-o-dsmt","8":"product_cat-o-dsmt-pellets","9":"product_cat-overig","10":"product_cat-pellets-for-pellet","11":"product_tag-nl","12":"product_tag-o-dsmt-ervaringen","13":"product_tag-o-dsmt","14":"product_tag-o-dsmt-bestellen","15":"product_tag-o-dsmt-kopen","16":"product_tag-o-dsmt-pellets","17":"product_tag-o-dsmt-psychonaut","18":"product_tag-o-dsmt-xl-pellets","19":"product_tag-what-is-o-dsmt","21":"first","22":"instock","23":"taxable","24":"shipping-taxable","25":"purchasable","26":"product-type-variable"},"_links":{"self":[{"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/product\/24864","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/comments?post=24864"}],"version-history":[{"count":5,"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/product\/24864\/revisions"}],"predecessor-version":[{"id":26437,"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/product\/24864\/revisions\/26437"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/media\/27932"}],"wp:attachment":[{"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/media?parent=24864"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/product_brand?post=24864"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/product_cat?post=24864"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/globalsourcechemicals.com\/et\/wp-json\/wp\/v2\/product_tag?post=24864"}],"curies":[{"name":"t\u00f6\u00f6leht","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}